Li-adrenoblock kapa li-adrenolytics ke lithethefatsi tse liehang kapa tse thibelang ho ba le maikutlo a mongobo, e.g. ba "tima" li-receptors tse ka marako a methapo ea mali le ka pelong, e sebetsang ho adrenaline le norepinephrine. Lethathamo la litokisetso - li-adrenoblock li ntse li eketseha selemo le selemo. A re ke re leke ho fumana hore na ke mofuta ofe oa li-adrenolytics tse teng, le hore na ke lintho life tseo ba sebetsang ka tsona.
Ke lithethefatsi tsa alpha le beta-li-adrenoblockers?
Mefuta e ka sehloohong ea adrenoblockers ke:
- alpha-blockers;
- beta-blockers.
Ho itšetlehile ka mofuta oa adrenolytics ho ama li-receptors tsa mofuta o mong oa mefuta e 'meli.
Li-adrenoblockers tse fapaneng li na le foromo e fapaneng ea tekanyo. Kahoo adrenolytics e tsoa ka foromo:
- matlapa;
- leboule le tharollo bakeng sa ente;
- marotholi.
Alpha receptor blockers
Li-alpha-adrenoblockers 'meleng li etsa lintho tse latelang:
- ho eketsa methapong e nyane, ha o ntse o fokotsa moroalo pelong;
- fokotsa khatello ea mocheso, ho fokotsa ho tsuba ha methapo ea mali le mojaro oa mesifa ea pelo;
- ntlafatsa ho potoloha ha mali;
- fokotsa khatello ho potoloho e nyane ea pulmona;
- k'holeseterole e tlase;
- fokotsa mahlaseli a tsoekere maling.
Sehlopha sa alpha-receptor blockers se kenyelletsa lithethefatsi tse sebelisoang ho latela lithethefatsi tse latelang:
- lefu la khatello ea mali;
- migraine ;
- lefu la endarteritis;
- sesebelisoa sa lijana tsa retinal.
Alfa-adrenoblockers e sebelisoa ka katleho phekolo e rarahaneng ea prostatitis ho banna.
Litlhaloso tse amanang le tšebeliso ea li-alpha-blockers ke mafu:
- hypotension e entsoeng ka matla;
- atherosclerosis;
- tšoaetso ea lik'hemik'hale;
- tšoaetso ea matšoao kapa ho se phekolehe hapatic.
Lethathamong la litokisetso tse tloaelehileng tsa alpha-blockers:
- Dihydroergotoxin;
- Urapidil;
- Nicergoline;
- Fentolamine;
- Pyrroxane;
- Tropafen;
- Prazosin hydrochloride;
- Butyroxane.
Bakeng sa tlhahisoleseding! Nakong e fetileng, lithethefatsi tse tsoang lethathamong la α-blocker li ne li sebelisetsoa ho hloekisa bakuli bohle ntle le khethollo, empa ka lebaka la lipatlisiso tsa bongaka li senotsoe hore ka linako tse ling kopo ea bona e ka lebisa ho hlasetsoeng ke pelo.
Beta-receptor blockers
Tsamaiso ea lithethefatsi tsa beta-blocker e lebisa ho phello e latelang:
- e fokotsa lebelo la pelo;
- e fokotsa khatello ea mali;
- ho hanyetsa ha lisele tsa pelo tsa mesifa ho ea ho oksijene tlala ea bo-'mchemia ho eketseha;
- ntlafatsa molumo oa methapo ea mali;
- ho thehoa ha thrombocyte ho thibetsoe;
- ho eketsa ho phalla ha oksijene likarong tsa 'mele;
- mosebetsi oa litho tsa ka hare le litšoelesa tsa sekhukhu li tsitsitse.
Lipontšo tsa tšebeliso ea lithethefatsi lethathamong la β-blockers ke mafu a kang:
- glaucoma;
- lefu la khatello ea mali;
- angina pectoris;
- pelo ea 'mele arrhythmia;
- tšoaetso ea lik'hemik'hale;
- ho hloleha ha pelo;
- thyrotoxicosis ;
- lefu la pelo.
Har'a li-contradiccation tse buang ka tšebeliso ea lithethefatsi tsa mofuta ona ke maloetse a 'maloa, ho akarelletsa:
- lefu la tsoekere;
- lefu la ho fokola ha pelo;
- COPD (boloetse bo sa foleng ba pulmonary disease);
- ho felisa atherosclerosis.
Lethathamong la beta-blockers ea moloko o mocha, lithethefatsi:
- Cordanum;
- Anaprilin (Propranolol);
- Metoprolol;
- Bisoprolol (Concor);
- Nebilet (Nebivolol);
- Betaxolol (Lokren);
- Aptin;
- Betazprin;
- Esmolol et al.
Bohlokoa! Le hoja lithethefatsi tse ling-li-adrenoblock li ka rekoa li-pharmacy tse se nang lengolo, empa li lokela ho sebelisoa ho ea ka ngaka ea ngaka, joalokaha litla-morao tse matla li ka fumanoa ho e-na le phekolo e nepahetseng.
Adrenoblockers ea motsoako
Ho na le sehlopha se khethehileng sa lithethefatsi tse iponahatsa ka nako e le 'ngoe e le li-alpha-adrenolytics le lithethefatsi tsa beta-adrenolytic. Tsena ke li-adrenoblockers, tse kang:
- Labetol;
- Procodolol.